Base-catalyzed synthesis of aryl amides from aryl azides and aldehydes
نویسندگان
چکیده
منابع مشابه
Synthesis of indolines, indoles, and benzopyrrolizidinones from simple aryl azides.
A simple approach to prepare indolines and benzopyrrolizidinones from ortho-azidoallylbenzenes via a tandem radical addition/cyclization is described. The use of triethylborane to initiate and sustain the process provides the best results. Indolines are easily converted into the corresponding indoles by oxidation with manganese dioxide.
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ژورنال
عنوان ژورنال: Chemical Science
سال: 2016
ISSN: 2041-6520,2041-6539
DOI: 10.1039/c5sc03510d